Olekšák, Patrik; Psotka, Miroslav; Vancurova, Marketa; Sapega, Olena; Bieblova, Jana; Reinis, Milan; Rysanek, David; Mikyskova, Romana; Chalupová, Katarína; Maliňák, Dávid; Svobodová, Jana; Andrýs, Rudolf; Řehulková, Helena; Škopek, Vojtěch; Pham, Ngoc Lam; Bartek, Jiri; Hodny, Zdenek; Musílek, Kamil
(Taylor & Francis, 2021)
Twelve novel analogs of STAT3 inhibitor BP-1-102 were designed and synthesised with the aim to modify hydrophobic fragments of the molecules that are important for interaction with the STAT3 SH2 domain. The cytotoxic ...