Jůza, Radomír; Stefkova, Kristyna; Dehaen, Wim; Randakova, Alena; Petrasek, Tomas; Vojtechova, Iveta; Kobrlova, Tereza; Pulkrabkova, Lenka; Muckova, Lubica; Mecava, Marko; Prchal, Lukas; Mezeiova, Eva; Musílek, Kamil; Soukup, Ondrej; Korabecny, Jan
(MDPI-Molecular diversity preservation international, 2021)
In this pilot study, a series of new 3,4-dihydroquinolin-2(1H)-one derivatives as potential dopamine receptor D-2 (D2R) modulators were synthesized and evaluated in vitro. The preliminary structure-activity relationship ...