Skok, Ziga; Barancokova, Michaela; Benek, Ondřej; Cruz, Cristina Durante; Tammela, Paivi; Tomasic, Tihomir; Zidar, Nace; Masic, Lucija Peterlin; Zega, Anamarija; Stevenson, Clare E. M; Mundy, Julia E. A; Lawson, David M; Maxwell, Anthony; Kikelj, Danijel; Ilas, Janez
(American chemical society, 2020)
We designed and synthesized a series of inhibitors of the bacterial enzymes DNA gyrase and DNA topoisomerase IV, based on our recently published benzothiazole-based inhibitor bearing an oxalyl moiety. To improve the ...